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4-Aroyl-3-hydroxy-5-phenyl-1H-pyrrol-2(5H)-ones as N-formyl peptide receptor 1 (FPR1) antagonists Journal article
BIOCHEMICAL PHARMACOLOGY, 2017,Volume: 142,Page: 120-132
Authors:  Kirpotina, Liliya N.;  Schepetkin, Igor A.;  Khlebnikov, Andrei I.;  Ruban, Olga I.;  Ge, Yunjun;  Ye, Richard D.;  Kominsky, Douglas J.;  Quinn, Mark T.
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Antagonist Formyl peptide receptor  1H-pyrrol-2(5H)-one  Neutrophil  Molecular modeling  
Synthesis of Five- and Six-Membered N-Phenylacetamido Substituted Heterocycles as Formyl Peptide Receptor Agonists Journal article
DRUG DEVELOPMENT RESEARCH, 2017,Volume: 78,Issue: 1,Page: 49-62
Authors:  Vergelli, Claudia;  Schepetkin, Igor A.;  Ciciani, Giovanna;  Cilibrizzi, Agostino;  Crocetti, Letizia;  Giovannoni, Maria Paola;  Guerrini, Gabriella;  Iacovone, Antonella;  Kirpotina, Liliya N.;  Ye, Richard D.;  Quinn, Mark T.
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formyl peptide receptor  agonist  pyridazin-3(2H)-one  neutrophil  Ca2+flux  
2-Arylacetamido-4-phenylamino-5-substituted pyridazinones as formyl peptide receptors agonists Journal article
Bioorganic and Medicinal Chemistry, 2016,Volume: 24,Issue: 11,Page: 2530-2543
Authors:  Vergelli C.;  Schepetkin I.A.;  Ciciani G.;  Cilibrizzi A.;  Crocetti L.;  Giovannoni M.P.;  Guerrini G.;  Iacovone A.;  Kirpotina L.N.;  Khlebnikov A.I.;  Ye R.D.;  Quinn M.T.
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Agonist  Ca2+ mobilization  Formyl peptide receptor (FPR)  Neutrophil  Pyridazin-3(2H)-one  
V101L of human formyl peptide receptor 1 (FPR1) increases receptor affinity and augments the antagonism mediated by cyclosporins Journal article
Biochemical Journal, 2013,Volume: 451,Issue: 2,Page: 245-255
Authors:  Zhou C.;  Zhou Y.;  Wang J.;  Feng Y.;  Wang H.;  Xue J.;  Chen Y.;  Ye R.D.;  Wang M.-W.
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Cyclosporin  Formyl peptide receptor 1 (FPR1)  Haplotype  Pharmacogenomics  Receptor affinity  Single nucleotide polymorphism  
Characterization of Quin-C1 for its anti-inflammatory property in a mouse model of bleomycin-induced lung injury Journal article
Acta Pharmacologica Sinica, 2011,Volume: 32,Issue: 5,Page: 601-610
Authors:  He M.;  Cheng N.;  Gao W.-W.;  Zhang M.;  Zhang Y.-Y.;  Ye R.D.;  Wang M.-W.
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anti-inflammation  bleomycin  cytokines  formyl peptide receptor  lung injury  Quin-C1  
Identification of functional domains in the formyl peptide receptor-like 1 for agonist-induced cell chemotaxis Journal article
FEBS Journal, 2005,Volume: 272,Issue: 3,Page: 769-778
Authors:  Le Y.;  Ye R.D.;  Gong W.;  Li J.;  Iribarren P.;  Wang J.M.
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Chemotaxis  Formyl peptide receptor  Formyl peptide receptor-like 1  Structure-function  
Novel chemoattractant peptides for human leukocytes Journal article
Biochemical Pharmacology, 2003,Volume: 66,Issue: 9,Page: 1841-1851
Authors:  Bae Y.-S.;  Park E.-Y.;  Kim Y.;  He R.;  Ye R.D.;  Kwak J.-Y.;  Suh P.-G.;  Ryu S.H.
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Chemotaxis  Formyl peptide receptor like 1  Peptide  Phagocytes  Phospholipase A2  Superoxide  
Characterization of chenodeoxycholic acid as an endogenous antagonist of the G-coupled formyl peptide receptors Journal article
Inflammation Research, 2000,Volume: 49,Issue: 12,Page: 744-755
Authors:  Chen X.;  Yang D.;  Shen W.;  Dong H.F.;  Wang J.M.;  Oppenheim J.J.;  Howard O.M.Z.
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Bile Acids  Chemotaxis  Chenodeoxycholic Acid  Formyl Peptide Receptor  Formyl Peptide Receptor Like 1. Calcium Flux  
The N-formyl peptide receptor: A model for the study of chemoattractant receptor structure and function Journal article
Pharmacology and Therapeutics, 1997,Volume: 74,Issue: 1,Page: 73-102
Authors:  Prossnitz E.R.;  Ye R.D.
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Chemoattractants  G-protein-coupled receptor  Inflammation  N-formyl peptide  N-formyl peptide receptor